Stephania Extract Cepharanthine Powder

Igama leMveliso: Stephania Japonica Extract
Imvelaphi yesiLatini: Stephania cephalantha Hayata(Stephania japonica (Thunb.) Miers)/ Stephania epigaea Lo/ Stephania yunnanensis HSLo.
Imbonakalo: Mhlophe, Grey Umgubo oMhlophe
Isithako esisebenzayo: Cepharanthine 80% -99% HPLC
Icandelo elisetyenzisiweyo: I-Tuber / Root
Isicelo: Iimveliso zezempilo
Indawo yokunyibilika: 145-155 °
Ukujikeleza okuthe ngqo: D20+277°(c=2inchloroform)
Indawo yokubila: 654.03°C (uqikelelo olurhabaxa)
Ubuninzi:1.1761(uqikelelo olurhabaxa)
Isalathiso seRefractive:1.5300(uqikelelo)
Iimeko zogcino:igesi engaphantsi (initrogen okanye iArgon) ku-2-8°C
Ukunyibilika: Ukunyibilika kwi-SO (35mg/mL) okanye i-ethanol (20mg/mL)
I-Acidity coefficient (pKa):7.61±0.20(Kuqikelelwe)


Iinkcukacha zeMveliso

Olunye ulwazi

Iithegi zeMveliso

Intshayelelo yeMveliso

I-Stephania Extract Cepharanthine Powder yinto ephuma kwimibhobho yesityalo i-Stephania cephalantha Hayata(Stephania japonica (Thunb.) Miers) okanye i-Stephania epigaea Lo/ Stephania yunnanensis HSLo.I-Cepharanthine yimveliso yendalo eyodwa kwesi sityalo kwaye ibe ngumxholo wezifundo ezahlukeneyo ngenxa yeempawu zayo ze-pharmacological.Ifunyaniswe ukuba ibonisa imisebenzi echasene ne-SARS-CoV-2, ebonisa impumelelo ekucinezeleni ukwanda kwentsholongwane.Ukongezelela, i-Cepharanthine ibonise ukukwazi ukuguqula i-P-glycoprotein (P-gp) -i-mediated multidrug resistance kwiiseli ezithile kunye nokuphucula uvakalelo lwe-anticancer agents kwiimodeli zokulinga.Ngaphezu koko, kuboniswe ukuba kuneempembelelo ezithintelayo kwi-cytochrome yesibindi somntu i-P450 enzymes CYP3A4, CYP2E1, kunye ne-CYP2C9, kwaye idibene ne-antitumor, i-anti-inflammatory, kunye ne-antinociceptive effects.
Isishwankathelo, i-Stephania Extract Cepharanthine Powder yifom yepowder yemveliso yendalo yeCepharanthine ephuma kwisityalo se-Stephania cephalantha, esibonise amandla kwizicelo ezahlukeneyo ze-pharmacological.

Inkcazo(COA)

Imveliso I-Cepharanthine
CAS 481-49-2
Isivavanyi 80%~99%
Imbonakalo Umgubo omhlophe
Ukupakisha I-1KG / Ibhegi yeFoil
Into Inkcazo
Imbonakalo umgubo ongwevu omhlophe, ivumba elingathathi hlangothi, i-hygroscopic kakhulu
Ukuchongwa I-TLC: Isisombululo esisemgangathweni kunye nesisombululo sovavanyo kwindawo efanayo, RF
Isivavanyi (isiseko esomileyo) 98.0%--102.0%
I-Specific Optical -2.4°~ -2.8°
PH 4.5~7.0
Iintsimbi ezinzima (NjengePb) ≤10ppm
As ≤1ppm
Pb ≤0.5ppm
Cd ≤1ppm
Hg ≤0.1ppm
Into enxulumeneyo Indawo ayikho nkulu kunendawo enesisombululo esisemgangathweni
Isinyibilikisi esishiyekileyo <0.5%
Umxholo wamanzi <2%

Iimpawu zeMveliso

I-Stephania Extract Cepharanthine Powder yimveliso yendalo ephuma kwisityalo uStephania cephalantha Hayata.Ifunyaniswe ineempawu ezininzi ze-pharmacological, kubandakanya:
1. Imisebenzi echasene ne-SARS-CoV-2
2. Iziphumo ezithintelayo ekwandeni kwentsholongwane egazini
3. Ukuguqulwa kwe-P-glycoprotein-mediated multidrug resistance
4. Ukomelezwa kovakalelo kwii-anticancer agents
5. Iziphumo ezithintelayo kwi-cytochrome yesibindi somntu i-P450 enzymes CYP3A4, CYP2E1, kunye ne-CYP2C9
6. I-Antitumor, i-anti-inflammatory, kunye ne-antinociceptive effects

Yintoni i-Biosynthesis yeCepharanthine?

I-biosynthesis ye-cepharanthine e-Stephania iqala nge-condensation ye-dopamine kunye ne-4-hydroxyphenylacetaldehyde (4-HPAA, i-5) nge-norcoclaurine synthase (NCS), i-norcoclaurine.

Yintoni i-Solubility yeCepharanthine?

I-Cepharanthine i-soluble kwii-solvents eziphilayo ezifana ne-ethanol, i-DMSO, kunye ne-dimethyl formamide (DMF).I-solubility ye-cepharanthine kula ma-solvents malunga ne-2, i-5, kunye ne-10 mg / ml, ngokulandelanayo.I-Cepharanthine iyanyibilika kancinane kwizithinteli ezinamanzi.

Usetyenziso

Imizi-mveliso yesicelo seStephania Extract Cepharanthine Powder ibandakanya iPharmaceutical, Nutraceutical, Biotechnology, kunye neHerbal Medicine, ezona zicelo ziphambili zezi zilandelayo:
Ukusetyenziswa okunokwenzeka kunyango lwe-antiviral
Okunokwenzeka njenge-adjuvant kunyango lomhlaza
Inokwenzeka ukuba isetyenziswe kunyango oluchasayo
Okunokwenzeka njenge-agent analgesic
Ezi zicelo zibonisa iindlela ezahlukeneyo zokusetyenziswa kweStephania Extract Cepharanthine Powder kwiimeko ezahlukeneyo zonyango.


  • Ngaphambili:
  • Okulandelayo:

  • Ukupakishwa kunye neNkonzo

    Ukupakishwa
    * Ixesha lokuhambisa: Malunga neentsuku ezi-3-5 zomsebenzi emva kwentlawulo yakho.
    * Iphakheji: Kwimigqomo yefiber eneeplastiki ezimbini ngaphakathi.
    * Ubunzima obuNina: 25kgs/idrum, Ubunzima obuGross: 28kgs/Drum
    * Ubungakanani beGubu kunye nomthamo: ID42cm × H52cm, 0.08 m³/ Igubu
    * Ugcino: Igcinwe kwindawo eyomileyo nepholileyo, zigcine kude nokukhanya okuqinileyo nobushushu.
    * Ubomi beShelf: Iminyaka emibini xa igcinwe kakuhle.

    Ukuhambisa ngenqanawe
    * I-DHL Express, i-FEDEX, kunye ne-EMS yobuninzi obungaphantsi kwe-50KG, edla ngokubizwa ngokuba yinkonzo ye-DDU.
    * Ukuthunyelwa kolwandle ngobuninzi obungaphezu kwe-500 kg;kunye nokuthunyelwa ngomoya kufumaneka kwi-50 kg ngaphezulu.
    * Kwiimveliso zexabiso eliphezulu, nceda ukhethe ukuthumela emoyeni kunye ne-DHL express ukhuseleko.
    * Nceda uqinisekise ukuba unako ukwenza imvume xa iimpahla zifikelela kumasiko akho ngaphambi kokufaka umyalelo.Kubathengi abavela eMexico, eTurkey, eItali, eRomania, eRashiya, nakwezinye iindawo ezikude.

    ukupakishwa kwe-bioway kwisicatshulwa sesityalo

    Iindlela zeNtlawulo kunye nokuhanjiswa

    Express
    Ngaphantsi kwe-100kg, iintsuku ezi-3-5
    Umnyango ukuya emnyango inkonzo lula ukuthatha iimpahla

    Ngaselwandle
    Ngaphezulu kwe-300kg, malunga neentsuku ezingama-30
    Izibuko ukuya kwinkonzo yezibuko umthengisi ovunyiweyo ofunekayo

    NgoMoya
    100kg-1000kg, 5-7 Iintsuku
    Isikhululo seenqwelomoya ukuya kwinkonzo yesikhululo seenqwelomoya siyafuneka

    utshintshe

    Iinkcukacha zeMveliso (Itshati yokuHamba)

    1. Ukufumana nokuVuna
    2. Ukutsalwa
    3. Ukugxila kunye nokuCoca
    4. Ukomisa
    5. Ukubekwa emgangathweni
    6. Ukulawulwa koMgangatho
    7. Ukupakishwa 8. Ukuhanjiswa

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