I-Stephania Extract Cepharanthine Powder

Igama leMveliso: I-Stephania Japonica Extract
Imvelaphi yesiLatini: Stephania cephalantha Hayata(Stephania japonica (Thunb.)Miers)/ Stephania epigaea Lo/ Stephania yunnanensis HSLo.
Inkangeleko: Mhlophe, uMpuphu oMhlophe ongwevu
Isithako Esisebenzayo: I-Cepharanthine 80%-99% HPLC
Icandelo elisetyenzisiweyo: I-Tuber/Root
Isicelo: Iimveliso zezeMpilo
Indawo yokunyibilika: 145-155°
Ujikelezo oluthile: D20+277°(c=2inchloroform)
Iqondo lokubila: 654.03°C (uqikelelo oluqikelelweyo)
Ubuninzi: 1.1761 (uqikelelo oluqikelelweyo)
Isalathisi sokubonisa ukukhanya: 1.5300 (uqikelelo)
Iimeko zokugcina: igesi ezingaphantsi komhlaba (initrogen okanye iArgon) kwi-2-8°C
Ukunyibilika: Inyibilika kwi-SO(35mg/mL) okanye kwi-ethanol(20mg/mL)
I-asidi efunekayo (pKa):7.61±0.20(Eqikelelweyo)


Iinkcukacha zeMveliso

Olunye ulwazi

Iithegi zeMveliso

Intshayelelo yeMveliso

I-Stephania Extract Cepharanthine Powder yinto ephuma kwiingcambu zesityalo i-Stephania cephalantha Hayata (Stephania japonica (Thunb.) Miers) okanye i-Stephania epigaea Lo/ Stephania yunnanensis HSLo. I-Cepharanthine yimveliso yendalo ehlukanisiweyo kwesi sityalo kwaye ibingumxholo wezifundo ezahlukeneyo ngenxa yeempawu zayo ezinokubakho ze-pharmacological. Kufunyenwe ukuba ibonisa imisebenzi yokulwa ne-SARS-CoV-2, ibonisa ukusebenza kakuhle ekuthinteleni ukwanda kwentsholongwane. Ukongeza, i-Cepharanthine ibonakalise amandla okuguqula ukumelana namayeza amaninzi okubangelwa yi-P-glycoprotein (P-gp) kwiiseli ezithile kwaye iphucula uvakalelo lweearhente zokulwa nomhlaza kwiimodeli zovavanyo. Ngaphezu koko, kubonakaliswe ukuba ineziphumo zokuthintela kwi-enzymes ze-cytochrome P450 zesibindi somntu i-CYP3A4, CYP2E1, kunye ne-CYP2C9, kwaye inxulunyaniswa neziphumo zokulwa nomhlaza, ukulwa nokuvuvukala, kunye ne-antinociceptive.
Ngamafutshane, iStephania Extract Cepharanthine Powder luhlobo lomgubo wemveliso yendalo iCepharanthine ephuma kwisityalo iStephania cephalantha, esibonakalise amandla kwiindlela ezahlukeneyo zokusetyenziswa kweyeza.

Inkcazo (i-COA)

Imveliso I-Cepharanthine
I-CAS 481-49-2
Uvavanyo 80%~99%
Inkangeleko Umgubo omhlophe
Ukupakisha Ingxowa ye-1KG/yeFoyile
Into Inkcazo
Inkangeleko umgubo omhlophe ongwevu, ivumba elingathathi cala, i-hygroscopic kakhulu
Ukuchongwa I-TLC: Isisombululo esiqhelekileyo kunye nesisombululo sovavanyo kwindawo enye, i-RF
Uvavanyo (Isiseko esomileyo) 98.0%--102.0%
I-Optical ethile -2.4°~ -2.8°
PH 4.5~7.0
Iintsimbi Ezinzima (Njenge-Pb) ≤10ppm
As ≤1ppm
Pb ≤0.5ppm
Cd ≤1ppm
Hg ≤0.1ppm
Izinto ezinxulumene noko Indawo engenkulu kunendawo yesisombululo esiqhelekileyo
Isinyibilikisi esiseleyo <0.5%
Umxholo wamanzi <2%

Iimpawu zeMveliso

I-Stephania Extract Cepharanthine Powder yimveliso yendalo ephuma kwisityalo i-Stephania cephalantha Hayata. Kufunyaniswe ukuba ineempawu ezininzi ze-pharmacological, kuquka:
1. Imisebenzi yokulwa ne-SARS-CoV-2
2. Imiphumo yokuthintela ukwanda kwentsholongwane
3. Ukuguqulwa kokumelana namayeza amaninzi okusetyenziswa yi-P-glycoprotein
4. Ukuphucula uvakalelo kwiiarhente zokulwa nomhlaza
5. Imiphumo yokuthintela kwi-enzymes ze-cytochrome P450 zesibindi somntu i-CYP3A4, i-CYP2E1, kunye ne-CYP2C9
6. Iziphumo zokulwa nomhlaza, ukudumba, kunye nokulwa nomhlaza

Yintoni i-Biosynthesis yeCepharanthine?

I-biosynthesis ye-cephalanthine eStephania iqala ngokudityaniswa kwe-dopamine kunye ne-4-hydroxyphenylacetaldehyde (4-HPAA, 5) nge-norcoclaurine synthase (NCS), nto leyo evelisa i-norcoclaurine.

Yintoni i-Solubility yeCepharanthine?

I-Cepharanthine iyanyibilika kwizinyibilikisi zendalo ezifana ne-ethanol, i-DMSO, kunye ne-dimethyl formamide (DMF). Ukunyibilika kwe-cepharanthine kwezi zinyibilikisi kumalunga ne-2, 5, kunye ne-10 mg/ml, ngokulandelelana. I-Cepharanthine ayinyibiliki kangako kwii-buffers zamanzi.

Izicelo

Amashishini asetyenziswa kwiStephania Extract Cepharanthine Powder aquka iPharmaceutical, Nutraceutical, Biotechnology, kunye neHerbal Medicine, izicelo eziphambili zezi zilandelayo:
Ukusetyenziswa okunokwenzeka kunyango lwe-antiviral
Isenokuba sisixhobo esincedisayo kunyango lomhlaza
Ingasetyenziswa kunyango lokulwa nokuvuvukala
Inokwenzeka njengeyeza lokuthomalalisa iintlungu
Ezi zicelo zibonisa iindlela ezahlukeneyo zokusetyenziswa kweStephania Extract Cepharanthine Powder kwiimeko ezahlukeneyo zonyango.


  • Ngaphambili:
  • Okulandelayo:

  • Ukupakishwa kunye neNkonzo

    Ukupakisha
    * Ixesha lokuHanjiswa: Malunga neentsuku ezi-3-5 zomsebenzi emva kwentlawulo yakho.
    * Iphakheji: Kwiidrum zefayibha kunye neengxowa ezimbini zeplastiki ngaphakathi.
    * Ubunzima obupheleleyo: 25kgs/igubu, Ubunzima obupheleleyo: 28kgs/igubu
    * Ubungakanani beDrum kunye nomthamo: ID42cm × H52cm, 0.08 m³/ Idrum
    * Indawo yokugcina: Igcinwe kwindawo eyomileyo nepholileyo, yigcine kude nokukhanya okunamandla nobushushu.
    * Ubomi beShelufu: Iminyaka emibini xa igcinwe kakuhle.

    Ukuhambisa ngenqanawe
    * I-DHL Express, i-FEDEX, kunye ne-EMS ngobuninzi obungaphantsi kwe-50KG, ngokuqhelekileyo ibizwa ngokuba yinkonzo ye-DDU.
    * Ukuthunyelwa ngenqanawa ngobuninzi obungaphezulu kwe-500 kg; kwaye ukuthunyelwa ngenqwelomoya kuyafumaneka nge-50 kg engaphezulu.
    * Kwiimveliso ezixabisa kakhulu, nceda ukhethe ukuthunyelwa ngenqwelo moya kunye ne-DHL express ukuze ukhuseleke.
    * Nceda uqinisekise ukuba unako na ukukhupha imvume xa iimpahla zifika kwi-customs yakho ngaphambi kokuba ufake i-odolo. Kubathengi abavela eMexico, eTurkey, e-Itali, eRomania, eRashiya, nakwezinye iindawo ezikude.

    iipakethi ze-bioway ze-extract yezityalo

    Iindlela zokuhlawula kunye nokuhambisa

    Express
    Ngaphantsi kwe-100kg, iintsuku ezi-3-5
    Inkonzo yokungena emnyango kulula ukuyithatha impahla

    Ngaselwandle
    Ngaphezulu kwe-300kg, malunga neentsuku ezingama-30
    Kufuneka umthengisi weenkonzo zokucoca iinqanawa ukusuka kwelinye izibuko ukuya kwelinye

    Ngomoya
    100kg-1000kg, iintsuku ezi-5-7
    Kufuneka umthengisi weenkonzo zokucoca izikhululo zeenqwelo-moya ukusuka kwisikhululo seenqwelo-moya ukuya kwisikhululo seenqwelo-moya

    utshintshiselwano

    Iinkcukacha zeMveliso (Itshati yokuHamba)

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